Description
Oleuropeinisabioactivecompoundfoundinallpartsoftheolivetree.OleuropeinhasbeenshowntoreduceintracellularROSgeneration,inhibitapoptosis,stABIlizemitochondrialmembranepotential,modulateapoptoticproteins,andincreasephosphorylationofAktandERK1/2inneonatalratcardiomyocytessubjectedtosimulationofischemia/reperfusion.Additionally,oleuropeinhasbeenfoundtodecreaseCOX-2expression,suppressIL-17inmucosaandsupernatant,andattenuateinflammatorydamageincolonicbiopsyculturesorsamplesofulcerativecolitis.FurThermore,oleuropeinwasfoundtosignificantlyincreaserADIosensitivityofnasopharyngealcarcinomacellsbyreducingexpressionofHIF1alpha,inadditiontoalteringexpressionsofmiRNAsandgenes.
References
ZhaoQ,BaiY,LiC,etal.Oleuropeinprotectscardiomyocyteagainstapoptosisviaactivatingthereperfusioninjurysalvagekinasepathwayinvitro.EvidBasedComplementAlternatMed.2017.2017:2109018.PMID:28491103.
LarussaT,OliverioM,SuraciE,etal.Oleuropeindecreasescyclooxygenase-2andinterleukin-17expressionandattenuatesinflammatorydamageincolonicsamplesfromulcerativecolitispatients.Nutrients.2017Apr15;9(4).pii:E391.PMID:28420140.
XuT,XiaoD.OleuropeinenhancesradiationsensitivityofnasopharyngealcarcinomabydownregulatingPDRG1throughHIF1alpha-repressedmicroRNA-519d.JExpClincancerRes.2017Jan5;36(1):3.PMID:28057028.
美国LKT Labs 是一家专注于防癌抗癌特殊化学品研究和开发的公司。主要提供:癌症药物、药物发现试剂盒、天然产物、广泛的生命科学研究试剂、定制合成。
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