品牌分类
品牌咨询
- CD4 Monoclonal Antibody (RM45), PE, eBioscience
- bpsbioscience常备现货
- 求教:BPS Bioscience官网 BPS Bioscience经销商/代理商,是假货吗?
- BPS bioscience代理_上海elisa生物技术有限公司
- GABAA Receptor β2 Subunit Polyclonal Antibody
- bpsbioscience抗体产品手机版
- 【Bpsbioscience代理】_上海酶联生物
- Antibodies, Proteins, Kits and Reagents for Life Science ...
- BRD4 (BD1) Inhibitor Screening Assay Kit性能参数,报价/价格,图片...
- BPS BioscienceELISA 试剂盒
- mysql源码安装_zengzehui的专栏
- BPS bioscience_BPS bioscience
联系方式
公司地址
苏州工业园区生物纳米园A4#216
联系电话
4000-520-616 / 18915418616
传真号码
0512-67156496
电子邮箱
info@ebiomall.com
公司网址
https://www.ebiomall.com
商品描述
MW:413.5Da
CASRegistry#:803712-79-0
Formula:C20H19N3O•CH4SO3
Description:
Obatoclax,alsoknownasGX15-070,isanovelBcl-2homologydomain-3(BH3)mimetic.ItoccupiesahydrophobiccleftwithintheBH3bindinggrooveofBcl-2,antagonizingBcl-2andthusinducingapoptosis.Obatoclaxinhibitedprimaryacutemyeloidleukemia(AML)ProgenitorcellproliferationwithanaverageIC50of0.18±0.07µM,anditpotentlyinducedapoptosisinprimaryAMLcellswithanaverageIC50of3.6±1.2µM.ObatoclaxovercomesBcl-2-,Bcl-xL-,Bcl-w-,andMcl-1-mediatedresistancetoBAXorBAKandtotheproteasomeinhibitorbortezomib.
Synonym(s):
GX15-070,Obatoclaxmesylate
Purity:
≥99%
Solubility:
SolubleinDMSOat5mg/ml;verypoorlysolubleinethanol;verypoorlysolubleinwater;maximumsolubilityinplainwaterisestimatedtobeabout200-400µM
Format:
Brownpowder
Storage/StABIlity:
Storeatorbelow–20°C.Solidformisstableatleast12monthsfromdateofreceipt,whenstoredasdirected.Donotstoreaqueoussolutionsformorethanoneday.
Reference(s):
1.Chonghaile,T.N.andLetai,A.Oncogene27:S149-S157(2008).
2.Konopleva,M.,etal.CancerRes.68:3413-3420(2008).
3.Nguyen,M.,etal.Proc.Natl.Acad.Sci.USA104:19512-19517(2007).
2.Konopleva,M.,etal.CancerRes.68:3413-3420(2008).
3.Nguyen,M.,etal.Proc.Natl.Acad.Sci.USA104:19512-19517(2007).
ScientificCategory:
Apoptosis
ProductType:
Inhibitor
Datashownislot-specific.Contactusforspecificinformationonotherlots.


