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联系方式
公司地址
苏州工业园区生物纳米园A4#216
联系电话
4000-520-616 / 18915418616
传真号码
0512-67156496
电子邮箱
info@ebiomall.com
公司网址
https://www.ebiomall.com
商品描述
MW:2091.5Da
Genbank#:NM_003548
Tag(s):none
a.a:1–21
Background:
Histoneacetyltransferase(HAT)p300/CBPcatalysestheacetylationofthisN-terminaltailoffreehistoneH4atLys5,8,12,16.Lys8isthoughttobethepreferredacetylationsiteinH4.Anumberofmethyltransferasesalsomodifythisregionofthehistone.
Description:
ApeptidesubstrateforHistone4R3methyltransferases.Thepeptidecorrespondstoaminoacidresidues1-21ofhistoneH4.
UniProt
P62805
Synonym(s):
H4,HIST4,Histoneh4
Purity:
≥95%byHPLC
SuppliedAs:
800µMsolutioninwater(200µl)
Format:
aqueoussolution
Storage/StABIlity:
≥ 12monthsat-20°Cor-70°C
Application(s):
Usefulasasubstrateforhistonemethyltransferase(atR3)andacetyltransferase(atK5,K8,K12andK16)familyassaysandforscreeningsmallmolecularinhibitorsofHistone4(R3)methyltransferasesfordrugdiscovery.
Reference(s):
ApplicationReference(s):
1.Differentialmodeofantimicrobialactionsofarginine-richandlysine-richhistonesagainstGram-positiveStaphylococcusaureus(2013)
2.ExtracellularhistonesareessentialeffectorsofC5aR-andC5L2-mediatedtissuedamageandinflammationinacutelunginjury(2013)
Warning(s):
Avoidfreeze/thawcycles.
AminoAcidSequence:
SGRGKGGKGLGKGGAKRHRKV
ScientificCategory:
Methyltransferase
ProductType:
Substrate
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