ubpbio/PYR-41/F5100/5 mg

价格
¥1500.00
货号:F5100
浏览量:127
品牌:UBPBio
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商品描述
PYR-41isacell-permeable,irreversIBLeubiquitin-activatingenzyme(E1)inhibitor(IC50<10=""μm).=""treatment=""of=""cells=""with=""pyr-41=""inhibits=""overall=""protein=""ubiquitination,=""prevents=""ubiquitin-mediated=""proteasomal=""degradation,=""and=""inhibits=""pathways=""mediated=""by=""the=""ubiquitin-proteasome.=""it=""has=""also=""been=""found=""that=""pyr-41=""treatment=""increases=""protein=""sumoylation=""in="">

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PYR-41isacell-permeable,irreversibleubiquitin-activatingenzyme(E1)inhibitor(IC50<10=""μm).=""treatment=""of=""cells=""with=""pyr-41=""inhibits=""overall=""protein=""ubiquitination,=""prevents=""ubiquitin-mediated=""proteasomal=""degradation,=""and=""inhibits=""pathways=""mediated=""by=""the=""ubiquitin-proteasome.=""it=""has=""also=""been=""found=""that=""pyr-41=""treatment=""increases=""protein=""sumoylation=""in=""cells.="">
Ubiquitin-Proteasome Biotechnologies成立于2011年,ubpbio是由科学家和投资者创立的私营企业。ubpbio致力于为学术界和工业界提供高质量的试剂和其他相关产品。ubpbio产品线包括的高度纯化的蛋白酶,E1和E2的酶,泛素和泛素衍生物,蛋白酶体抑制剂和蛋白酶基板。ubpbio不断开发创新以增加新的产品,ubpbio致力为全球的客户提供更多的帮助。在人类细胞中,有超过1000的蛋白质/酶,参与维持泛素-蛋白酶体系统的正常活动。失调的UPS已发现涉及大量的人类疾病包括癌症的病理生理,炎性疾病和神经退行性疾病。ubpbio致力为客户提供更好的泛素-蛋白酶体系统解决方案。
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ProductName:PYR-41
AlsoKnownAs:4[4-(5-Nitro-furan-2-ylmethylene)-3,5-dioxo-pyrazolidin-1-yl]-benzoicacidethylester
CatalogNo.:F5100
Size:5mg
MolecularWeight:371.3Da
Species:N/A
Source:Synthetic
Stock:Powder
Concentration:N/A
QualityAssurance:>98%(TLC);NMR(Confirms)
Storage:Eligibleforroomtemperatureshipping.Storeat-20°Cuponreceiving;protectfromairandlight
PDFDataSheet:PDFDatasheet
NCBIRefSeq:N/A
Image(s):N/A
ShippingMethod:Roomtemperatureshipping
References:Yang,Y.,etal.(2007)CancerRes.67:9472.